SCHEMBL9301537

SCHEMBL9301537

COC1CCOC(c2cc(O)cc(F)c2)C1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 2/20 0.35
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9268003 0.80 CA12 (0.36) DRD3CA12CA1CA9
SCHEMBL6024905 0.79 DRD3 (0.50) DRD3
SCHEMBL8410875 0.74 HCAR1 (0.32) DRD3CA12CA1CA9
SCHEMBL28806180 0.69 CYP19A1 (0.32) CA12CA1CA9
SCHEMBL14721136 0.69 SLC6A4 (0.37)
SCHEMBL9159765 0.69 HTR2C (0.40) DRD3
SCHEMBL9300450 0.67 TLR9 (0.32)
SCHEMBL9157877 0.65 DRD3 (0.32) DRD3
SCHEMBL9159596 0.65 DRD3 (0.32) DRD3
SCHEMBL7532624 0.64 CA12 (0.43) CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5308852-A Cardiovascular disorders MERCK FROSST CANADA, INC. (CA) 1994-05-03 US disclosed
EP-0579304-A1 Heteroarylnaphthalenes as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1994-01-19 EP disclosed
WO-1994000444-A1 HETEROARYLNAPHTHALENES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1994-01-06 WO disclosed
EP-0375404-A2 Heterocyclic derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-27 EP disclosed