SCHEMBL9301558

SCHEMBL9301558

CCOC(=O)Cc1cncc(C#Cc2cc3c(cc2C)SCCC3(C)C)n1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RARA P10276 8/20 0.46
RARB P10826 8/20 0.46
RARG P13631 8/20 0.46
KMT2A Q03164 3/20 0.46
CYP3A4 P08684 2/20 0.46
CYP26A1 O43174 1/20 0.37
MEN1 O00255 2/20 0.31
RXRA P19793 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
RXRB P28702 1/20 0.30
RXRG P48443 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302053 0.89 CYP3A4 (0.43) RARARARBRARGKMT2ACYP3A4
SCHEMBL9302702 0.89 RARA (0.41) RARARARBRARGKMT2ACYP3A4
SCHEMBL9303919 0.86 RARA (0.64) RARARARBRARGKMT2ACYP3A4
SCHEMBL9302684 0.82 RARA (0.46) RARARARBRARGKMT2ACYP3A4
SCHEMBL9304096 0.81 RARA (0.51) RARARARBRARGKMT2ACYP3A4
SCHEMBL9302090 0.81 RARA (0.39) RARARARBRARGKMT2ACYP3A4
SCHEMBL9302065 0.81 RARA (0.44) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817713 0.79 RARA (0.49) RARARARBRARGKMT2ACYP3A4
SCHEMBL6668128 0.78 RARA (0.48) RARARARBRARGKMT2ACYP3A4
SCHEMBL8658232 0.78 CYP3A4 (0.41) RARARARBRARGKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed