SCHEMBL9303919

SCHEMBL9303919

CCOC(=O)Cc1cncc(C#Cc2ccc3c(c2)C(C)(C)CCS3)n1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RARA P10276 11/20 0.64
RARB P10826 11/20 0.64
RARG P13631 11/20 0.64
KMT2A Q03164 4/20 0.64
CYP3A4 P08684 3/20 0.64
CYP26A1 O43174 2/20 0.54
RXRA P19793 2/20 0.36
CRABP2 P29373 1/20 0.33
MEN1 O00255 3/20 0.32
CSF1R P07333 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303289 0.89 RARA (0.59) RARARARBRARGKMT2ACYP3A4
SCHEMBL9302591 0.88 RARB (0.61) RARARARBRARGKMT2ACYP3A4
SCHEMBL9301558 0.86 RARA (0.46) RARARARBRARGKMT2ACYP3A4
SCHEMBL9303234 0.84 RARB (0.61) RARARARBRARGKMT2ACYP3A4
SCHEMBL9302658 0.83 RARB (0.67) RARARARBRARGKMT2ACYP3A4
SCHEMBL9304071 0.82 RARA (0.44) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817758 0.81 RARA (0.62) RARARARBRARGKMT2ACYP3A4
SCHEMBL9303296 0.81 RARA (0.60) RARARARBRARGKMT2ACYP3A4
SCHEMBL9301486 0.80 RARB (0.56) RARARARBRARGKMT2ACYP3A4
SCHEMBL19342930 0.79 RARA (0.78) RARARARBRARGKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed