SCHEMBL9301967

SCHEMBL9301967

COC(=O)[C@H](Cc1ccccc1)NC(=O)CC(N)C(=O)O

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.58
KLK5 Q9Y337 1/20 0.57
ALDH1A1 P00352 3/20 0.56
THRB P10828 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
HSD17B10 Q99714 1/20 0.56
POLB P06746 1/20 0.55
LMNA P02545 2/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
GLA P06280 1/20 0.53
HDAC1 Q13547 3/20 0.53
HDAC6 Q9UBN7 3/20 0.53
MDM4 O15151 1/20 0.53
MDM2 Q00987 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8603038 1.00 ATM (0.58) ATMKLK5ALDH1A1THRBCYP2C9
SCHEMBL11406714 1.00 ATM (0.58) ATMKLK5ALDH1A1THRBCYP2C9
SCHEMBL6549557 1.00 ATM (0.58) ATMKLK5ALDH1A1THRBCYP2C9
Hydrochloric Acid SCHEMBL9492789 0.99 ATM (0.56) ATMKLK5ALDH1A1THRBCYP2C9
SCHEMBL8603938 0.93 ATM (0.59) ATMKLK5ALDH1A1THRBCYP2C9
SCHEMBL8603937 0.93 ATM (0.59) ATMKLK5ALDH1A1THRBCYP2C9
Hydrochloric Acid SCHEMBL10412319 0.92 ATM (0.58) ATMKLK5ALDH1A1THRBCYP2C9
SCHEMBL8086148 0.92 ALDH1A1 (0.55) ATMKLK5ALDH1A1THRBCYP2C9
SCHEMBL237136 0.89 ACE (0.57) ATMKLK5
SCHEMBL22013341 0.89 ATM (0.60) ATMKLK5ALDH1A1THRBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334236-B1 Preparation of n-protected alpha-l-aspartyl-l-phenylalanine methyl ester MITSUI TOATSU CHEMICALS (JP) 1994-08-31 EP disclosed
US-5302743-A Reacting N-protected L-aspartic anhydride with L-phenylalanine methyl ester salt in non-aqueous solvent MITSUI TOATSU CHEMICALS, INC. (JP) 1994-04-12 US disclosed
US-4549987-A DEFORMYLATION AND SEPARATION OF N-FORMYL-L-A-ASPARTYL-L-PHENYLALANINE METHYL ESTER FARMITALIA CARLO ERBA S.P.A. (IT) 1985-10-29 US disclosed