SCHEMBL9302019

SCHEMBL9302019

CCCC(C(=O)OCC)c1ncc(C#Cc2cc3c(cc2C)SCCC3(C)C)cn1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.47
RARA P10276 2/20 0.47
RARB P10826 2/20 0.47
RARG P13631 2/20 0.47
KMT2A Q03164 1/20 0.47
CYP26A1 O43174 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302216 0.91 RARA (0.43) CYP3A4RARARARBRARGKMT2A
SCHEMBL9817829 0.86 RARB (0.47) CYP3A4RARARARBRARGKMT2A
SCHEMBL9303664 0.85 CYP3A4 (0.44) CYP3A4RARARARBRARGKMT2A
SCHEMBL9304096 0.83 RARA (0.51) CYP3A4RARARARBRARGKMT2A
SCHEMBL9302770 0.82 RXRA (0.37) CYP3A4RARARARBRARGKMT2A
SCHEMBL9302065 0.82 RARA (0.44) CYP3A4RARARARBRARGKMT2A
SCHEMBL6667776 0.79 RARA (0.47) CYP3A4RARARARBRARGKMT2A
SCHEMBL9817823 0.79 RARB (0.47) CYP3A4RARARARBRARGKMT2A
SCHEMBL6664858 0.78 CYP26A1 (0.46) CYP3A4RARARARBRARGKMT2A
SCHEMBL9302613 0.78 CYP3A4 (0.39) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed