SCHEMBL9302758

SCHEMBL9302758

Cc1cc2c(cc1C#Cc1cnc(CCCCC(=O)O)nc1)C(C)(C)CCO2

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 5/20 0.38
RXRA P19793 2/20 0.36
HNF4A P41235 1/20 0.36
CYP26A1 O43174 2/20 0.34
CYP26B1 Q9NR63 2/20 0.34
PTGER4 P35408 8/20 0.34
RARA P10276 3/20 0.33
RARB P10826 3/20 0.33
RARG P13631 3/20 0.33
S1PR5 Q9H228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6671507 0.89 RXRA (0.37) FFAR1RXRAHNF4ARARARARB
SCHEMBL6664727 0.87 CYP26A1 (0.40) FFAR1RXRAHNF4ACYP26A1CYP26B1
SCHEMBL9303121 0.85 RXRA (0.34) FFAR1RXRAHNF4ACYP26A1CYP26B1
SCHEMBL9301731 0.85 CYP26A1 (0.41) RXRAHNF4ACYP26A1CYP26B1PTGER4
SCHEMBL9139409 0.85 RXRA (0.37) FFAR1RXRAHNF4ARARARARB
SCHEMBL9139432 0.84 RXRA (0.34) FFAR1RXRAHNF4ACYP26A1CYP26B1
SCHEMBL6669202 0.81 RXRA (0.37) RXRAHNF4ARARARARBRARG
SCHEMBL9302221 0.81 CYP3A4 (0.43) FFAR1RXRACYP26A1CYP26B1RARA
SCHEMBL7649079 0.81 TBXAS1 (0.31) RARARARBRARG
SCHEMBL9301379 0.80 RXRA (0.40) RXRAHNF4ACYP26A1CYP26B1RARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed