SCHEMBL9302941

SCHEMBL9302941

CCCC(C(=O)OCC)c1cc(C#Cc2ccc3c(c2)C(C)(C)CCO3)cnn1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RARB P10826 7/20 0.39
RARG P13631 7/20 0.39
RARA P10276 6/20 0.39
CYP3A4 P08684 2/20 0.39
KMT2A Q03164 1/20 0.39
RXRA P19793 2/20 0.35
HNF4A P41235 1/20 0.35
CYP26A1 O43174 2/20 0.33
CYP26B1 Q9NR63 1/20 0.33
CRABP2 P29373 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303529 0.90 RARB (0.38) RARBRARGRARACYP3A4KMT2A
SCHEMBL9301695 0.88 RXRA (0.34) RARBRARGRARACYP3A4KMT2A
SCHEMBL9303163 0.85 RARB (0.43) RARBRARGRARACYP3A4KMT2A
SCHEMBL9304047 0.85 RARA (0.42) RARBRARGRARACYP3A4KMT2A
SCHEMBL9302111 0.83 RARB (0.57) RARBRARGRARACYP3A4KMT2A
SCHEMBL9303176 0.80 RARB (0.41) RARBRARGRARACYP3A4KMT2A
SCHEMBL9303114 0.79 RXRA (0.33) RARBRARGRARARXRAHNF4A
SCHEMBL9302931 0.77 RARA (0.39) RARBRARGRARACYP3A4KMT2A
SCHEMBL9301727 0.77 RARB (0.39) RARBRARGRARACYP3A4KMT2A
SCHEMBL9304352 0.75 CYP26A1 (0.46) RARBRARGRARACYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed