SCHEMBL9303069

SCHEMBL9303069

COC(=O)OS(=O)(=O)Cc1ccc([N+](=O)[O-])cc1.[NaH]

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.48
HTT P42858 1/20 0.48
GAA P10253 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 3/20 0.43
F2 P00734 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HTR2A P28223 1/20 0.43
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872160 0.83 HTT (0.51) POLBHTTGAAMAPTKMT2A
SCHEMBL27485980 0.80 KMT2A (0.49) MAPTKMT2AALDH1A1F2PRSS1
SCHEMBL22163994 0.79 KMT2A (0.48) POLBHTTGAAMAPTKMT2A
SCHEMBL28498471 0.79 HTT (0.57) POLBHTTKMT2AALDH1A1TSHR
SCHEMBL27519584 0.78 KMT2A (0.50) MAPTKMT2AALDH1A1F2PRSS1
SCHEMBL11722467 0.77 GAA (0.54) POLBHTTGAAMAPTKMT2A
Hydrochloric Acid SCHEMBL27483889 0.76 KMT2A (0.49) MAPTKMT2AALDH1A1F2PRSS1
SCHEMBL8078609 0.75 HTT (0.57) POLBHTTGAAMAPTKMT2A
SCHEMBL6141208 0.75 HTR2A (0.64) HTTGAAMAPTALDH1A1RAB9A
SCHEMBL1425402 0.74 LOXL2 (0.57) POLBHTTGAAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360802-A Antagonists of cholecystokinin and gastrin MERCK SHARPE & DOHME LTD. 1994-11-01 US disclosed
EP-0514133-A1 Benzodiazepine derivatives, compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1992-11-19 EP disclosed