SCHEMBL9304008

SCHEMBL9304008

NC(=O)c1ccc2[nH]c(Cl)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 18/20 0.49
PKN1 Q16512 1/20 0.44
PKN2 Q16513 1/20 0.44
MEN1 O00255 1/20 0.44
THRB P10828 1/20 0.44
KMT2A Q03164 1/20 0.44
MMP2 P08253 1/20 0.43
MMP13 P45452 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304016 0.87 CHEK2 (0.63) CHEK2PKN1PKN2MEN1THRB
SCHEMBL13836654 0.86 CHEK2 (0.47) CHEK2MEN1THRBKMT2A
SCHEMBL30167005 0.85 TDP1 (0.49) CHEK2MEN1THRBKMT2A
SCHEMBL9928725 0.85 TDP1 (0.49) CHEK2MEN1THRBKMT2A
SCHEMBL22121440 0.81 FABP6 (0.51) CHEK2PKN1PKN2MEN1KMT2A
SCHEMBL18745926 0.81 CHEK2 (0.47) CHEK2PKN1PKN2KMT2AMMP2
SCHEMBL30732472 0.81 CHEK2 (0.47) CHEK2PKN1PKN2MMP2MMP13
SCHEMBL16318609 0.80 CHEK2 (0.49) CHEK2PKN1PKN2MMP2MMP13
SCHEMBL8262964 0.80 HSP90AA1 (0.55) CHEK2PKN1PKN2KMT2AMMP2
SCHEMBL16134556 0.80 CHEK2 (0.46) CHEK2PKN1PKN2MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed