SCHEMBL9304540

SCHEMBL9304540

CCCCCCc1ccc2nc(S)[nH]c2c1Br

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.35
TYR P14679 2/20 0.35
CYP3A4 P08684 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
ALOX5 P09917 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TLR8 Q9NR97 5/20 0.34
KDM4E B2RXH2 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29094812 0.84 PTGS2 (0.38) KCNH2TYRCYP3A4MAPTMEN1
SCHEMBL9306904 0.83 KCNH2 (0.35) KCNH2TYRCYP3A4MAPTMEN1
SCHEMBL31332112 0.83 TLR8 (0.41) CYP3A4MAPTTLR8KDM4EUSP2
SCHEMBL27654237 0.80 TLR8 (0.44) KCNH2TLR8LIPG
SCHEMBL9304517 0.78 KCNH2 (0.35) KCNH2TYRCYP3A4MAPTMEN1
SCHEMBL9847103 0.70 TYR (0.43) KCNH2TYRCYP3A4MAPTMEN1
SCHEMBL9305967 0.69 S1PR4 (0.60) TSHRTLR8S1PR4S1PR1S1PR5
SCHEMBL28208703 0.68 TYR (0.47) KCNH2TYRCYP3A4MAPTMEN1
SCHEMBL11615877 0.67 TYR (0.46) KCNH2TYRCYP3A4MAPTMEN1
SCHEMBL11616253 0.67 TYR (0.46) KCNH2TYRCYP3A4MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0161220-B1 PROCESS FOR THE PREPARATION OF BETA-(BENZOTHIAZOLYLTHIO) AND BETA (BENZIMIDAZOLYLTHIO)CARBOXYLIC-ACID DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-14 EP disclosed
US-4652653-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio)-carboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1987-03-24 US disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed