SCHEMBL9304517

SCHEMBL9304517

CCCCCCc1ccc2[nH]c(S)nc2c1Br

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.35
TYR P14679 2/20 0.35
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX5 P09917 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HSD17B10 Q99714 1/20 0.33
LIPG Q9Y5X9 1/20 0.33
GPR84 Q9NQS5 3/20 0.31
TLR8 Q9NR97 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9306899 0.83 NPC1 (0.38) KCNH2TYRMEN1TP53CYP3A4
SCHEMBL9304540 0.78 KCNH2 (0.35) KCNH2TYRMEN1TP53CYP3A4
SCHEMBL9305320 0.72 TYR (0.38) KCNH2TYRMEN1TP53CYP3A4
SCHEMBL9305489 0.72 KCNH2 (0.35) KCNH2TYRMEN1TP53CYP3A4
SCHEMBL9847100 0.70 TYR (0.43) KCNH2TYRMEN1TP53CYP3A4
SCHEMBL9305960 0.69 S1PR4 (0.47) TP53CYP3A4HSD17B10TLR8
SCHEMBL28208703 0.68 TYR (0.47) KCNH2TYRMEN1TP53CYP3A4
SCHEMBL29094812 0.68 PTGS2 (0.38) KCNH2TYRMEN1TP53CYP3A4
SCHEMBL9306904 0.67 KCNH2 (0.35) KCNH2TYRMEN1TP53CYP3A4
SCHEMBL9305443 0.67 ALDH1A1 (0.40) KCNH2TYRMEN1TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0161220-B1 PROCESS FOR THE PREPARATION OF BETA-(BENZOTHIAZOLYLTHIO) AND BETA (BENZIMIDAZOLYLTHIO)CARBOXYLIC-ACID DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-14 EP disclosed
US-4652653-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio)-carboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1987-03-24 US disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed
EP-0161220-A2 Process for the preparation of beta-(benzothiazolylthio) and beta (benzimidazolylthio)carboxylic-acid derivatives CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed
EP-0126030-A2 Process for the preparation of beta-(benzothiazolylthio) and beta-(benzimidazolylthio) carboxylic acids CIBA-GEIGY AG (CH) 1984-11-21 EP disclosed