SCHEMBL9304760

SCHEMBL9304760

NCCNCc1cc(Br)no1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.34
MC5R P33032 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
NOTUM Q6P988 2/20 0.32
IGF1R P08069 1/20 0.32
CA12 O43570 2/20 0.31
CA6 P23280 2/20 0.31
CA7 P43166 2/20 0.31
CA9 Q16790 2/20 0.31
CA14 Q9ULX7 2/20 0.31
CA5B Q9Y2D0 2/20 0.31
MEN1 O00255 1/20 0.31
RECQL P46063 1/20 0.31
KMT2A Q03164 1/20 0.31
CHRM1 P11229 1/20 0.30
ALDH1A1 P00352 2/20 0.30
LMNA P02545 2/20 0.30
TDP1 Q9NUW8 2/20 0.30
JAK2 O60674 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10863100 0.80 MC4R (0.35) MC4RMC5RHRH3CA12CA6
SCHEMBL7992705 0.79 VHL (0.41) MC4RMC5RHRH3IGF1RMEN1
SCHEMBL10862922 0.79 MC4R (0.34) MC4RMC5RHRH3CA12CA6
SCHEMBL10865896 0.79 SIGMAR1 (0.34) MC4RMC5RHRH3NOTUMCA12
SCHEMBL10862013 0.78 HRH3 (0.47) MC4RMC5RHRH3CHRM1ALDH1A1
SCHEMBL10864820 0.76 EPHX2 (0.43) MC4RMC5RHRH3IGF1RKMT2A
SCHEMBL10864880 0.76 HRH3 (0.34) MC4RMC5RHRH3ALDH1A1JAK2
SCHEMBL10864502 0.75 EPHX2 (0.44) MC4RMC5RIGF1RALDH1A1LMNA
SCHEMBL10865941 0.75 CACNA1G (0.32) MC4RMC5RHRH3
SCHEMBL10863059 0.75 MC4R (0.32) MC4RMC5RHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360906-A N-(3-halo-5-isoxazolylmethyl)-2-nitromethylene- and -2-nitroimino-imidazolines and pyrimidines; aminoalkylation, cyclization SHELL RESEARCH LIMITED (GB) 1994-11-01 US disclosed
EP-0555931-A1 Isoxazole derivatives and their use as pesticides SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1993-08-18 EP disclosed
EP-0192060-A1 Heterocyclic compounds NIHON BAYER AGROCHEM K.K. (JP) 1986-08-27 EP disclosed