SCHEMBL9305342

SCHEMBL9305342

O=C(O)CC(C(O)=S)c1nc2c(-c3ccccc3)cccc2o1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.39
CTSA P10619 11/20 0.38
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
CASP1 P29466 1/20 0.34
MMP12 P39900 1/20 0.34
MMP13 P45452 1/20 0.34
LIPG Q9Y5X9 1/20 0.34
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9305331 0.90 TOP2A (0.36) TOP2ACTSAPIK3CDPIK3CAPIK3CB
SCHEMBL9306240 0.82 DAGLA (0.42) CTSAPIK3CDPIK3CBMMP12MMP13
SCHEMBL9305328 0.81 TOP2A (0.40) TOP2APIK3CDPIK3CAPIK3CBLIPG
SCHEMBL8973089 0.81 IKBKE (0.35) CTSA
SCHEMBL8972338 0.80 HDAC3 (0.46)
SCHEMBL9304112 0.80 CTSA (0.33) CTSA
SCHEMBL9733965 0.80 CTSA (0.33) CTSA
Ammonia Solution, Strong SCHEMBL10865678 0.79 HDAC3 (0.45)
SCHEMBL9306352 0.78 HSD17B10 (0.37)
Methylamine SCHEMBL10867855 0.77 HDAC4 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
US-4612049-A BENZOTHI ZOLYL THIO-, BENZIMIDAZOLYLTHIO- OR BENZOXAZOLYLTHIO-SUBSTITUTED CARBOXY ACID CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed