SCHEMBL9305844

SCHEMBL9305844

O=C(S)CC(C(=O)O)c1nc2cc(C(F)(F)F)ccc2s1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.48
AKR1B1 P15121 16/20 0.47
AKR1A1 P14550 5/20 0.43
ALOX5 P09917 1/20 0.42
AKR1B10 O60218 1/20 0.40
GLO1 Q04760 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
NCS1 P62166 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9305859 0.82 AKR1B1 (0.49) DYRK1AAKR1B1AKR1A1ALOX5AKR1B10
SCHEMBL8972937 0.81 NPC1 (0.54) DYRK1ATRPV1
SCHEMBL8972523 0.81 DYRK1A (0.46) DYRK1AAKR1B1
SCHEMBL8973355 0.81 PPARA (0.50) AKR1B1ALOX5
SCHEMBL9443356 0.79 NPC1 (0.42) DYRK1AALOX5TRPV1
SCHEMBL9305849 0.79 DYRK1A (0.43) DYRK1AAKR1B1AKR1A1ALOX5AKR1B10
SCHEMBL9443094 0.79 DYRK1A (0.54) DYRK1AAKR1B1AKR1A1ALOX5TRPV1
SCHEMBL9304878 0.78 NPC1 (0.55) DYRK1A
SCHEMBL9443201 0.78 ALDH1A1 (0.41) ALOX5TRPV1
SCHEMBL9306659 0.78 PPARA (0.47) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0375614-B1 CORROSION-INHIBITING COATING COMPOSITIONS CIBA-GEIGY AG (CH) 1993-03-31 EP disclosed
US-5198482-A Benzothiazole carboxylic acid amine salt CIBA-GEIGY CORPORATION (US) 1993-03-30 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0375614-A1 Corrosion-inhibiting coating compositions CIBA-GEIGY AG (CH) 1990-06-27 EP disclosed
US-4612049-A BENZOTHI ZOLYL THIO-, BENZIMIDAZOLYLTHIO- OR BENZOXAZOLYLTHIO-SUBSTITUTED CARBOXY ACID CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed