SCHEMBL9305859

SCHEMBL9305859

O=C(O)CC(C(O)=S)c1nc2cc(C(F)(F)F)ccc2s1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 17/20 0.49
DYRK1A Q13627 1/20 0.47
AKR1A1 P14550 5/20 0.47
AKR1B10 O60218 1/20 0.44
GLO1 Q04760 1/20 0.44
TRPV1 Q8NER1 1/20 0.42
ALOX5 P09917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9305849 0.90 DYRK1A (0.43) AKR1B1DYRK1AAKR1A1AKR1B10GLO1
SCHEMBL9305844 0.82 DYRK1A (0.48) AKR1B1DYRK1AAKR1A1AKR1B10GLO1
SCHEMBL8972535 0.81 DYRK1A (0.45) AKR1B1DYRK1AAKR1A1TRPV1
SCHEMBL8972967 0.81 NPC1 (0.52) TRPV1
SCHEMBL8973369 0.81 HDAC6 (0.55) AKR1B1ALOX5
SCHEMBL9443373 0.80 NPC1 (0.41) DYRK1ATRPV1
SCHEMBL9443106 0.79 DYRK1A (0.49) AKR1B1DYRK1AAKR1A1TRPV1ALOX5
SCHEMBL9304897 0.79 NPC1 (0.54) AKR1B1DYRK1A
SCHEMBL9306671 0.79 PPARA (0.46) DYRK1A
SCHEMBL9443212 0.79 ALDH1A1 (0.43) AKR1B1TRPV1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0375614-B1 CORROSION-INHIBITING COATING COMPOSITIONS CIBA-GEIGY AG (CH) 1993-03-31 EP disclosed
US-5198482-A Benzothiazole carboxylic acid amine salt CIBA-GEIGY CORPORATION (US) 1993-03-30 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0375614-A1 Corrosion-inhibiting coating compositions CIBA-GEIGY AG (CH) 1990-06-27 EP disclosed
US-4612049-A BENZOTHI ZOLYL THIO-, BENZIMIDAZOLYLTHIO- OR BENZOXAZOLYLTHIO-SUBSTITUTED CARBOXY ACID CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed