SCHEMBL9305928

SCHEMBL9305928

CC(C)Oc1ccc2nc(S)[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 1/20 0.56
PDE3B Q13370 1/20 0.49
PDE3A Q14432 1/20 0.49
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CYP1A2 P05177 7/20 0.46
CYP2E1 P05181 7/20 0.46
CYP3A4 P08684 7/20 0.46
CYP2C8 P10632 7/20 0.46
CYP2D6 P10635 7/20 0.46
CYP2C9 P11712 7/20 0.46
CYP2B6 P20813 7/20 0.46
CYP2C19 P33261 7/20 0.46
PTPRC P08575 1/20 0.44
PTPRF P10586 1/20 0.44
PTPN2 P17706 1/20 0.44
PTPN1 P18031 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9305942 0.87 PDE3B (0.46) CBFBPDE3BPDE3AHDAC3HDAC1
SCHEMBL2108226 0.84 CYP3A4 (0.49) CBFBCYP1A2CYP2E1CYP3A4CYP2C8
SCHEMBL916533 0.81 NPC1 (0.58) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL29770426 0.81 NPC1 (0.58) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL9305034 0.81 CBFB (0.56) CBFBPDE3BPDE3AHDAC3HDAC1
SCHEMBL9148442 0.80 NPC1 (0.56) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
Hydrochloric Acid SCHEMBL28679041 0.80 NPC1 (0.56) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL26189984 0.78 NPC1 (0.40) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL16208344 0.78 RAB9A (0.49) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL4591067 0.77 NPC1 (0.47) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0161220-B1 PROCESS FOR THE PREPARATION OF BETA-(BENZOTHIAZOLYLTHIO) AND BETA (BENZIMIDAZOLYLTHIO)CARBOXYLIC-ACID DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-14 EP disclosed
US-4652653-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio)-carboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1987-03-24 US disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed
EP-0161220-A2 Process for the preparation of beta-(benzothiazolylthio) and beta (benzimidazolylthio)carboxylic-acid derivatives CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed
EP-0126030-A2 Process for the preparation of beta-(benzothiazolylthio) and beta-(benzimidazolylthio) carboxylic acids CIBA-GEIGY AG (CH) 1984-11-21 EP disclosed