SCHEMBL9305034

SCHEMBL9305034

CC(C)Oc1ccc2nc(Cl)[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 1/20 0.56
PDE3B Q13370 1/20 0.49
PDE3A Q14432 1/20 0.49
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
PTPRC P08575 1/20 0.46
PTPRF P10586 1/20 0.46
PTPN2 P17706 1/20 0.46
PTPN1 P18031 1/20 0.46
CYP1A2 P05177 7/20 0.46
CYP2E1 P05181 7/20 0.46
CYP3A4 P08684 7/20 0.46
CYP2C8 P10632 7/20 0.46
CYP2D6 P10635 7/20 0.46
CYP2C9 P11712 7/20 0.46
CYP2B6 P20813 7/20 0.46
CYP2C19 P33261 7/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9305044 0.87 PDE3B (0.46) CBFBPDE3BPDE3AHDAC3HDAC1
SCHEMBL3140572 0.83 ALDH1A1 (0.46) PDE3BPDE3AHDAC3HDAC1HDAC2
SCHEMBL1748047 0.81 NPC1 (0.58) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL9305928 0.81 CBFB (0.56) CBFBPDE3BPDE3AHDAC3HDAC1
SCHEMBL9304850 0.77 NPC1 (0.61) CBFBPDE3BPDE3ACYP1A2CYP2E1
SCHEMBL2728712 0.75 SCN10A (0.55) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL32674484 0.74 RUNX1 (0.56) CBFBCYP1A2CYP3A4CYP2C9NPC1
SCHEMBL13219327 0.74 RUNX1 (0.56) CBFBCYP1A2CYP3A4CYP2C9NPC1
SCHEMBL24553690 0.74 CBFB (0.49) CBFBPDE3BPDE3AHDAC3HDAC1
SCHEMBL15647884 0.73 MEN1 (0.57) CBFBPDE3BPDE3AHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed