SCHEMBL9306154

SCHEMBL9306154

CC(C)(C)c1cccc2nc(Br)sc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.39
GABRA1 P14867 1/20 0.34
GABRB2 P47870 1/20 0.34
CASR P41180 2/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
PLA2G1B P04054 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TNF P01375 1/20 0.33
NOD1 Q9Y239 1/20 0.33
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24820021 0.83 HDAC3 (0.44) ALDH1A1HDAC3HDAC4HDAC1HDAC7
SCHEMBL13305137 0.81 RAB9A (0.41) CA2GABRA1GABRB2CASRALDH1A1
SCHEMBL9305633 0.79 CA2 (0.38) CA2GABRA1GABRB2CASRALDH1A1
SCHEMBL19226220 0.79 CA2 (0.38) CA2GABRA1GABRB2CASRALDH1A1
SCHEMBL23421550 0.79 ASH1L (0.42) CA2ALDH1A1MAPTTSHRTDP1
SCHEMBL11831944 0.78 KMT2A (0.42) CA2CASRALDH1A1TSHRTDP1
SCHEMBL18791158 0.72 PSMB8 (0.58) ALDH1A1MAPTTDP1HDAC3HDAC4
SCHEMBL31389941 0.72 PSMB8 (0.37) ALDH1A1MAPTTDP1PSMB8
SCHEMBL19008541 0.72 CA2 (0.38) CA2GABRA1GABRB2CASRALDH1A1
SCHEMBL12829698 0.72 HDAC3 (0.41) CASRALDH1A1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0129506-B1 HETEROCYCLICALLY SUBSTITUTED THIO(CYCLO)ALKANE POLYCARBOXYLIC ACIDS CIBA-GEIGY AG (CH) 1991-03-06 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed