SCHEMBL9306380

SCHEMBL9306380

COc1cc(O)cc2nc(S)[nH]c12

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
ESR2 Q92731 5/20 0.39
ESR1 P03372 4/20 0.39
PTGS2 P35354 2/20 0.37
ALOX5 P09917 1/20 0.37
MAOB P27338 1/20 0.35
PDE4A P27815 1/20 0.34
PDE4D Q08499 1/20 0.34
SMPD3 Q9NY59 3/20 0.33
AMY1A P0DUB6 3/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
FLT3 P36888 1/20 0.32
NOX1 Q9Y5S8 1/20 0.32
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16198229 0.80 AMY1A (0.36) MAPTAMY1AKDM4EALDH1A1
SCHEMBL9306577 0.80 ESR2 (0.42) CYP3A4MAPTESR2ESR1PTGS2
SCHEMBL7479166 0.78 CYP3A4 (0.39) CYP3A4MAPTESR2ESR1PTGS2
SCHEMBL9306374 0.73 CYP3A4 (0.41) CYP3A4MAPTESR2ESR1PTGS2
SCHEMBL2549634 0.72 NQO2 (0.44) MAPTAMY1AKDM4EALDH1A1LMNA
SCHEMBL21723167 0.69 MAPT (0.52) CYP3A4MAPTESR2ESR1PTGS2
SCHEMBL211457 0.68 AMY1A (0.45) ALOX5AMY1APDGFRBPDGFRA
SCHEMBL23757778 0.67 CYP3A4 (0.61) CYP3A4MAPTESR2ESR1PTGS2
SCHEMBL8064768 0.66 CYP3A4 (0.67) CYP3A4MAPTESR2ESR1PTGS2
SCHEMBL9455942 0.64 AMY1A (0.47) MAPTALOX5AMY1AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed