SCHEMBL9307958

SCHEMBL9307958

Cc1cc2oc(=O)c(NC(=O)C(F)c3ccc(F)cc3)c(-c3ccccc3C)c2cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.39
THRB P10828 1/20 0.39
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ESR1 P03372 2/20 0.37
ESR2 Q92731 1/20 0.37
LMNA P02545 2/20 0.36
MAPT P10636 4/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
HTR1E P28566 1/20 0.35
S1PR3 Q99500 1/20 0.35
MAOB P27338 2/20 0.35
MAOA P21397 1/20 0.34
TDP1 Q9NUW8 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9155117 0.82 NPC1 (0.42) NPC1RAB9AHTTSMN1; SMN2
SCHEMBL9153940 0.81 MAOB (0.43) TP53KDM4EHPGDALDH1A1GAA
SCHEMBL9307949 0.79 TP53 (0.39) TP53KDM4EHPGDALDH1A1GAA
SCHEMBL9150777 0.74 SMN1; SMN2 (0.45) KDM4EALDH1A1LMNAMAPTMEN1
SCHEMBL9154464 0.73 KDR (0.48) TP53LMNAMAPTMEN1KMT2A
SCHEMBL9153164 0.72 KDM4E (0.38) TP53KDM4EHPGDALDH1A1GAA
SCHEMBL6940744 0.72 NPC1 (0.42) NPC1RAB9AHTTSMN1; SMN2
SCHEMBL9154452 0.71 RECQL (0.46) KDM4EALDH1A1NPC1RAB9AHTT
SCHEMBL9158313 0.71
SCHEMBL9153131 0.70 CYP1A2 (0.43) TP53KDM4EHPGDALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5278186-A Substituted with secondary amide TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-01-11 US disclosed