SCHEMBL9308045

SCHEMBL9308045

O=C1OC(=O)c2cc3ncccc3cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.47
POLB P06746 3/20 0.47
RAB9A P51151 1/20 0.47
PDGFRB P09619 1/20 0.46
PDGFRA P16234 1/20 0.46
CASP6 P55212 1/20 0.44
ALDH1A1 P00352 6/20 0.44
HTT P42858 5/20 0.44
TP53 P04637 3/20 0.44
MAPT P10636 3/20 0.44
CASP1 P29466 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 2/20 0.44
HSP90AA1 P07900 2/20 0.44
TSHR P16473 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CASP7 P55210 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5393255 0.83 POLB (0.46) NPC1POLBRAB9APDGFRBPDGFRA
SCHEMBL2936414 0.79 TDP1 (0.42) NPC1RAB9AALDH1A1MAPTMEN1
SCHEMBL20062355 0.78 ALDH1A1 (0.54) NPC1POLBRAB9APDGFRBPDGFRA
SCHEMBL29350099 0.76 NPC1 (0.65) NPC1POLBRAB9APDGFRBPDGFRA
SCHEMBL150476 0.76 NPC1 (0.65) NPC1POLBRAB9APDGFRBPDGFRA
SCHEMBL6647315 0.74 NPC1 (0.62) NPC1POLBRAB9APDGFRBPDGFRA
SCHEMBL30083328 0.74 ALOX15 (0.60) POLBRAB9AALDH1A1HTTTP53
SCHEMBL103 0.74 ALOX15 (0.60) POLBRAB9AALDH1A1HTTTP53
SCHEMBL21187608 0.73 ALDH1A1 (0.57) NPC1POLBRAB9APDGFRBPDGFRA
SCHEMBL13495403 0.73 PDGFRB (0.50) NPC1POLBRAB9APDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4622967-A1 COMPOUNDS THAT INHIBIT PKMYT1 Exelixis, Inc. (US) 2025-10-01 EP disclosed
WO-2024112853-A1 COMPOUNDS THAT INHIBIT PKMYT1 EXELIXIS, INC. (US) 2024-05-30 WO disclosed
WO-2024112853-A1 COMPOUNDS THAT INHIBIT PKMYT1 EXELIXIS, INC. (US) 2024-05-30 WO disclosed
US-5283335-A Controlling (mono or di)cotyledenous plants AMERICAN CYANAMID COMPANY (US) 1994-02-01 US disclosed