SCHEMBL9310772

SCHEMBL9310772

COc1c(C)c(C)c(OC)c(C(CCCO)c2ccccc2)c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.36
HRH1 P35367 3/20 0.36
TBXA2R P21731 1/20 0.36
CYP2C9 P11712 3/20 0.34
TRPA1 O75762 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
GSR P00390 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
BRD4 O60885 1/20 0.32
BRD2 P25440 1/20 0.32
BRD3 Q15059 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9310154 0.94 TBXA2R (0.39) HTR2AHRH1TBXA2RCYP2C9TRPA1
SCHEMBL9308785 0.94 TBXA2R (0.39) HTR2AHRH1TBXA2RCYP2C9TRPA1
SCHEMBL9307887 0.94 TBXA2R (0.39) HTR2AHRH1TBXA2RCYP2C9TRPA1
SCHEMBL9309778 0.87 TBXA2R (0.38) HTR2AHRH1TBXA2RCYP2C9TRPA1
SCHEMBL9662366 0.87 SIGMAR1 (0.38) HTR2AHRH1TBXA2RCYP2C9SIGMAR1
SCHEMBL9310821 0.87 HRH1 (0.37) HTR2AHRH1TBXA2RCYP2C9SIGMAR1
SCHEMBL9308823 0.86 TBXA2R (0.39) HTR2AHRH1TBXA2RCYP2C9TRPA1
SCHEMBL9549814 0.86 TBXAS1 (0.41) PDE4D
SCHEMBL9310439 0.86 TBXA2R (0.34) HTR2AHRH1TBXA2RCYP2C9SIGMAR1
SCHEMBL10866141 0.85 SIGMAR1 (0.41) HTR2AHRH1TBXA2RCYP2C9SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304658-A Quinone derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-04-19 US disclosed
US-5180742-A Lipoxygenase Inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-19 US disclosed
EP-0171251-B2 QUINONE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-12-23 EP disclosed
EP-0171251-B1 QUINONE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1990-06-27 EP disclosed
EP-0171251-A2 Quinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1986-02-12 EP disclosed