SCHEMBL9311982

SCHEMBL9311982

Cc1cccc(-c2ccccc2)c1NC(N)=S

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
TP53 P04637 1/20 0.44
TYR P14679 1/20 0.44
TSHR P16473 1/20 0.44
TAS2R38 P59533 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MAPT P10636 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GAA P10253 2/20 0.41
CYP1A2 P05177 2/20 0.41
POLB P06746 2/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX12 P18054 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 2/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9060479 0.82 POLB (0.45) ALDH1A1MAPTGAACYP1A2POLB
SCHEMBL5222474 0.82 GRIN2D (0.55) ALDH1A1MAPTL3MBTL1GAACYP1A2
SCHEMBL9537883 0.80 CYP2A6 (0.47) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL9539998 0.80 ALDH1A1 (0.44) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL9311503 0.78 EPHX1 (0.62) ALDH1A1MAPTL3MBTL1GAACYP1A2
SCHEMBL28726710 0.78 ALDH1A1 (0.42) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL9537505 0.77 SLC9A1 (0.42) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL18509790 0.74 ESR2 (0.42) ALDH1A1TSHRHSD17B10CYP1A2POLB
SCHEMBL16351359 0.74 ALDH1A1 (0.47) ALDH1A1TSHRMAPTHTTSMN1; SMN2
SCHEMBL9059999 0.74 SMN1; SMN2 (0.39) ALDH1A1TSHRMAPTL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536151-B1 ORTHOSUBSTITUTED BIPHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM BOOTS CO PLC (GB) 1994-09-14 EP disclosed
US-5302720-A Biphenyl-substituted guanidine derivatives useful as hypoglycaemic agents THE BOOTS COMPANY (GB) 1994-04-12 US disclosed
EP-0536151-A1 ORTHOSUBSTITUTED BIPHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM. BOOTS CO PLC (GB) 1993-04-14 EP disclosed
WO-1992000273-A1 ORTHOSUBSTITUTED BIPHENYL AMIDINE AND BIPHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM THE BOOTS COMPANY PLC (GB) 1992-01-09 WO disclosed