SCHEMBL931248

SCHEMBL931248

COc1ccc(C2(c3cccc(-c4cncnc4)c3)N=C(N)c3nccnc32)cc1C1CC1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.53
BACE2 Q9Y5Z0 8/20 0.53
CTSD P07339 6/20 0.53
KCNH2 Q12809 8/20 0.49
REN P00797 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3357414 0.89 BACE1 (0.54) BACE1BACE2CTSDKCNH2REN
SCHEMBL6885096 0.88 BACE1 (0.51) BACE1BACE2CTSDKCNH2REN
SCHEMBL6887443 0.84 BACE1 (0.42) BACE1BACE2CTSDKCNH2REN
SCHEMBL930937 0.82 BACE1 (0.67) BACE1BACE2KCNH2
SCHEMBL931345 0.82 BACE1 (0.67) BACE1BACE2KCNH2
SCHEMBL931386 0.82 BACE1 (0.67) BACE1BACE2KCNH2
SCHEMBL29767725 0.81 BACE1 (0.61) BACE1BACE2CTSDKCNH2REN
SCHEMBL931362 0.81 BACE1 (0.61) BACE1BACE2CTSDKCNH2REN
SCHEMBL931249 0.79 BACE1 (0.45) BACE1BACE2CTSDKCNH2REN
SCHEMBL3358057 0.78 BACE1 (0.51) BACE1BACE2CTSDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO disclosed