SCHEMBL9315657

SCHEMBL9315657

Cc1noc(-c2cccc(NC(=O)O)c2)n1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.64
MAPT P10636 2/20 0.64
POLB P06746 1/20 0.64
HAVCR2 Q8TDQ0 6/20 0.53
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
TSHR P16473 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
CA2 P00918 1/20 0.48
KIF18A Q8NI77 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.46
MAPK10 P53779 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31362862 0.79 NR1H4 (0.69) TP53MAPTPOLBNPC1RAB9A
SCHEMBL24247776 0.79 BRD4 (0.57) TP53MAPTPOLBNPC1RAB9A
SCHEMBL940686 0.79 NR1H4 (0.69) TP53MAPTPOLBNPC1RAB9A
SCHEMBL13415304 0.79 TP53 (0.64) TP53MAPTNPC1RAB9ATSHR
SCHEMBL4456834 0.79 TP53 (0.62) TP53MAPTPOLBHAVCR2NPC1
SCHEMBL27631838 0.79 TP53 (0.49) TP53MAPTPOLBHAVCR2NPC1
SCHEMBL9414015 0.77 MAPT (0.52) TP53MAPTPOLBHAVCR2NPC1
SCHEMBL9315056 0.75 MAPT (0.48) TP53MAPTPOLBHAVCR2NPC1
SCHEMBL860042 0.75 TP53 (0.56) TP53MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL12494 0.75 RAB9A (0.64) TP53MAPTPOLBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5374643-A Aryl urea (thiourea) and cyanoguanidine derivatives E. R. SQUIBB & SONS, INC. (US) 1994-12-20 US disclosed
EP-0587180-A2 Aryl urea (Thiourea) and cyanoguanidine derivatives E.R. SQUIBB & SONS, INC. (US) 1994-03-16 EP disclosed