SCHEMBL931589

SCHEMBL931589

CC1=NC(c2c(C#N)ccc(F)c2-c2ccccc2O)(C2CC2)N=C1N

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.40
KCNH2 Q12809 5/20 0.40
BACE2 Q9Y5Z0 2/20 0.38
APP P05067 8/20 0.36
IKBKB O14920 1/20 0.32
PGR P06401 2/20 0.32
AR P10275 2/20 0.32
CHUK O15111 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL976638 0.71 BACE1 (0.56) BACE1KCNH2BACE2APP
SCHEMBL6891149 0.67 BACE1 (0.58) BACE1KCNH2BACE2APP
SCHEMBL932719 0.66 BACE1 (0.57) BACE1KCNH2BACE2APP
SCHEMBL932326 0.65 BACE1 (0.56) BACE1KCNH2BACE2APP
SCHEMBL25006211 0.61 MEN1 (0.49)
SCHEMBL932205 0.61 BACE1 (0.61) BACE1KCNH2BACE2APP
SCHEMBL931600 0.60 BACE1 (0.55) BACE1KCNH2BACE2APP
SCHEMBL29403248 0.59 ESR2 (0.52) PGRARCHUK
SCHEMBL6752587 0.59 ESR2 (0.52) PGRARCHUK
SCHEMBL31589804 0.59 ALDH1A1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed