SCHEMBL932326

SCHEMBL932326

COc1cccc(-c2cc(C3(C4CC4)N=C(C)C(N)=N3)ccc2O)c1F

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.56
KCNH2 Q12809 5/20 0.52
APP P05067 4/20 0.46
BACE2 Q9Y5Z0 2/20 0.43
PFKFB3 Q16875 1/20 0.35
CTSD P07339 1/20 0.35
KDM1A O60341 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931135 0.81 BACE1 (0.52) BACE1KCNH2APPBACE2CTSD
SCHEMBL6891149 0.79 BACE1 (0.58) BACE1KCNH2APPBACE2
SCHEMBL932719 0.78 BACE1 (0.57) BACE1KCNH2APPBACE2CTSD
SCHEMBL931425 0.77 BACE1 (0.52) BACE1KCNH2APPBACE2KDM1A
SCHEMBL976638 0.74 BACE1 (0.56) BACE1KCNH2APPBACE2KDM1A
SCHEMBL931601 0.73 BACE1 (0.50) BACE1KCNH2APPBACE2
SCHEMBL931600 0.73 BACE1 (0.55) BACE1KCNH2APPBACE2
SCHEMBL1075789 0.72 BACE1 (0.74) BACE1KCNH2APPBACE2
SCHEMBL931611 0.71 BACE1 (0.68) BACE1KCNH2BACE2
SCHEMBL932236 0.70 BACE1 (0.53) BACE1KCNH2APPBACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO claimed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed