SCHEMBL9316190

SCHEMBL9316190

COc1cc(OC)nc(NC(=O)NS(=O)(=O)Nc2ccc(C(=O)C3CC3)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
CDK1 P06493 1/20 0.46
CYP1A2 P05177 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPT P10636 2/20 0.39
TP53 P04637 1/20 0.39
GLA P06280 1/20 0.39
ALOX15 P16050 1/20 0.39
CHIA Q9BZP6 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
KCNH2 Q12809 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
POLB P06746 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
GFER P55789 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9316966 0.85 GAA (0.50) GAACDK1CYP1A2ALDH1A1MAPT
SCHEMBL53468 0.82 GAA (0.47) GAACDK1CYP1A2ALDH1A1MAPT
SCHEMBL29510603 0.82 GAA (0.47) GAACDK1CYP1A2ALDH1A1MAPT
SCHEMBL6812884 0.81 GAA (0.47) GAACDK1CYP1A2ALDH1A1MAPT
SCHEMBL8539345 0.80 GAA (0.45) GAACDK1CYP1A2ALDH1A1MAPT
SCHEMBL8539307 0.79 GAA (0.44) GAACDK1CYP1A2ALDH1A1MAPT
SCHEMBL6573975 0.79 GAA (0.54) GAACDK1CYP1A2ALDH1A1MAPT
SCHEMBL8859618 0.79 GAA (0.60) GAACDK1CYP1A2ALDH1A1MAPT
SCHEMBL10948960 0.78 GAA (0.52) GAACDK1CYP1A2MAPTTP53
SCHEMBL8534941 0.77 GAA (0.49) GAACDK1CYP1A2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5280007-A Using 1-(a,a-dimethylbenzyl)-3-p-tolyurea and s-(1-methyl-1-phenylethyl-1-piperidinecarbothioate AMERICAN CYANAMID COMPANY (US) 1994-01-18 US claimed