SCHEMBL9316491

SCHEMBL9316491

CC12CC3CC(C)(C1)CC(NC(=N)Nc1ccccc1I)(C3)C2.Cc1ccccc1NC(=N)NC12CC3CC(C)(CC(C)(C3)C1)C2

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.51
GRIN2D O15399 5/20 0.51
GRIN3B O60391 5/20 0.51
GRIN1 Q05586 5/20 0.51
GRIN2A Q12879 5/20 0.51
GRIN2B Q13224 5/20 0.51
GRIN2C Q14957 5/20 0.51
GRIN3A Q8TCU5 5/20 0.51
EPHX2 P34913 12/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6720587 0.94 SIGMAR1 (0.56) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6720873 0.93 EPHX2 (0.55) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL28396308 0.79 EPHX2 (0.76) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6158255 0.77 SIGMAR1 (0.53) SIGMAR1EPHX2
SCHEMBL6155754 0.77 SIGMAR1 (0.55) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL8874234 0.76 SIGMAR1 (0.54) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8996696 0.75 SIGMAR1 (0.60) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6719463 0.75 SIGMAR1 (0.51) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
Guanidine SCHEMBL9516168 0.73 SIGMAR1 (0.56) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9316511 0.70 EPHX2 (0.44) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532642-A4 1994-04-27 EP claimed
EP-0532642-A1 SUBSTITUTED GUANIDINES HAVING HIGH BINDING TO THE SIGMA RECEPTOR AND THE USE THEREOF STATE OF OREGON, acting through OREGON STATE BOARD OF HIGHER EDUCATION, acting for OREGON HEALTH SC. UNIV. AND UNIV. OF OREGON (US) 1993-03-24 EP claimed
WO-1991018868-A1 SUBSTITUTED GUANIDINES HAVING HIGH BINDING TO THE SIGMA RECEPTOR AND THE USE THEREOF STATE OF OREGON, acting by and through the OREGON STATE BOARD OF HIGHER EDUCATION, acting for and onbehalf of the OREGON HEALTH SCIENCES UNIVERSITY (US) 1991-12-12 WO claimed