SCHEMBL9317643

SCHEMBL9317643

CC(N)C(OCc1cc(Br)cc(Br)c1)(c1ccccc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.46
IDO1 P14902 1/20 0.39
EDNRB P24530 1/20 0.35
EDNRA P25101 1/20 0.35
CACNA1F O60840 1/20 0.34
CACNA1D Q01668 1/20 0.34
CACNA1S Q13698 1/20 0.34
CACNA1C Q13936 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9318573 0.85 TACR1 (0.49) TACR1IDO1EDNRBEDNRA
SCHEMBL8460283 0.84 TACR1 (0.50) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9317784 0.81 TACR1 (0.58) TACR1IDO1CACNA1FCACNA1DCACNA1S
SCHEMBL9319570 0.81 TACR1 (0.45) TACR1EDNRBEDNRA
SCHEMBL9392799 0.81 TACR1 (0.58) TACR1IDO1CACNA1FCACNA1DCACNA1S
SCHEMBL9318574 0.79 TACR1 (0.47) TACR1EDNRBEDNRA
SCHEMBL9318203 0.77 PNMT (0.50) TACR1IDO1
SCHEMBL9318544 0.74 GLA (0.43) TACR1
SCHEMBL9318581 0.73 TACR1 (0.50) TACR1EDNRBEDNRACACNA1FCACNA1D
SCHEMBL9318137 0.72 RAB9A (0.46) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593557-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY. MERCK SHARP & DOHME (GB) 1994-04-27 EP claimed
EP-0593557-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY. MERCK SHARP & DOHME (GB) 1994-04-27 EP disclosed