SCHEMBL9320604

SCHEMBL9320604

CNc1ccc(C(=O)N2CCN(CCc3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.68
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
KCNH2 Q12809 1/20 0.56
DRD3 P35462 2/20 0.56
GPR183 P32249 1/20 0.55
LSS P48449 1/20 0.55
POLB P06746 1/20 0.55
HTR2A P28223 1/20 0.55
DRD2 P14416 2/20 0.52
KCNA5 P22460 2/20 0.52
LMNA P02545 1/20 0.51
HPGD P15428 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9426784 0.99 THRB (0.67) THRBKDM4EALDH1A1MAPTMEN1
SCHEMBL9513241 0.90 THRB (0.82) THRBKDM4EALDH1A1MAPTMEN1
Dimethylamine SCHEMBL9320437 0.89 THRB (0.63) THRBKDM4EALDH1A1MAPTMEN1
SCHEMBL9320194 0.88 THRB (0.65) THRBKDM4EALDH1A1MAPTMEN1
SCHEMBL9319893 0.88 THRB (0.65) THRBKDM4EALDH1A1MAPTMEN1
SCHEMBL9426220 0.88 MEN1 (0.56) MEN1KMT2AKCNH2HTR2A
SCHEMBL9320357 0.88 THRB (0.68) THRBMEN1KMT2AKCNH2GPR183
SCHEMBL9426171 0.86 THRB (0.63) THRBKDM4EALDH1A1MAPTMEN1
SCHEMBL9512997 0.86 THRB (0.73) THRBKDM4EALDH1A1MAPTMEN1
SCHEMBL10898714 0.86 THRB (0.73) THRBKDM4EALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5321027-A Analgesic CIBA-GEIGY CORPORATION (US) 1994-06-14 US disclosed
US-5286728-A Amino-substituted piperazine derivatives CIBA-GEIGY CORPORATION (US) 1994-02-15 US disclosed
EP-0524146-A1 Aminosubstituted Piperazinederivatives CIBA-GEIGY AG (CH) 1993-01-20 EP disclosed
EP-0489690-A1 Substituted N-Benzoyl-N'-(2-phenylethyl)-piperazines CIBA-GEIGY AG (CH) 1992-06-10 EP disclosed