SCHEMBL9323970

SCHEMBL9323970

CC(OS(C)(=O)=O)c1ccc2ccccc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP1A2 P05177 2/20 0.39
PTGS2 P35354 1/20 0.38
KDM4E B2RXH2 2/20 0.38
PRNP P04156 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
RXFP1 Q9HBX9 2/20 0.38
MAPK10 P53779 1/20 0.38
NCF1 P14598 3/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HPGD P15428 1/20 0.36
S1PR3 Q99500 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5797187 0.80 CYP1A2 (0.46) ALDH1A1HSD17B10CYP1A2PTGS2KDM4E
SCHEMBL31373891 0.78 CYP1A2 (0.45) ALDH1A1HSD17B10CYP1A2KDM4EPRNP
SCHEMBL28308791 0.78 CYP1A2 (0.45) ALDH1A1HSD17B10CYP1A2KDM4EPRNP
SCHEMBL9400811 0.75 ALDH1A1 (0.47) ALDH1A1HSD17B10CYP1A2PTGS2KDM4E
SCHEMBL20023734 0.74 CYP1A2 (0.44) ALDH1A1CYP1A2KDM4EKMT2ALMNA
SCHEMBL506970 0.73 HTT (0.41) ALDH1A1HSD17B10KDM4ELMNAHTT
SCHEMBL506969 0.73 HTT (0.41) ALDH1A1HSD17B10KDM4ELMNAHTT
SCHEMBL1713701 0.73 UGT2B7 (0.50) CYP1A2KMT2ACA9
SCHEMBL1261380 0.73 CYP1A2 (0.48) ALDH1A1HSD17B10CYP1A2KDM4EPRNP
SCHEMBL827081 0.73 CYP1A2 (0.52) ALDH1A1HSD17B10CYP1A2KDM4EPRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5334719-A Antihistamines, antiallergens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1994-08-02 US disclosed
US-5298512-A Substituted chromans and their use in the treatment of asthma, arthritis and related diseases PFIZER INC. (US) 1994-03-29 US disclosed
EP-0391625-B1 Substituted chromans in the treatment of asthma, arthritis and related diseases PFIZER (US) 1994-01-26 EP disclosed
WO-1993025546-A1 BICYCLIC(AZAAROMATIC)INDOLES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1993-12-23 WO disclosed
EP-0391625-A1 Substituted chromans in the treatment of asthma, arthritis and related diseases PFIZER INC. (US) 1990-10-10 EP disclosed