SCHEMBL932215

SCHEMBL932215

CSC1=NC(c2ccc(OC(F)F)cc2)(c2cccc(Br)c2)N=C1N

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.41
REN P00797 3/20 0.39
CTSD P07339 3/20 0.39
BACE2 Q9Y5Z0 3/20 0.39
KCNH2 Q12809 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932184 0.86 BACE1 (0.48) BACE1CTSDBACE2KCNH2
SCHEMBL932844 0.85 BACE1 (0.50) BACE1RENCTSDBACE2KCNH2
SCHEMBL932646 0.84 BACE1 (0.46) BACE1CTSDKCNH2
SCHEMBL932551 0.83 BACE1 (0.40) BACE1RENCTSDBACE2KCNH2
SCHEMBL932513 0.76 BACE1 (0.51) BACE1CTSDBACE2KCNH2
SCHEMBL947178 0.75 CTSD (0.37) BACE1CTSDBACE2
SCHEMBL932202 0.74 BACE1 (0.34) BACE1CTSDBACE2
SCHEMBL932175 0.71 BACE1 (0.51) BACE1CTSDBACE2KCNH2
SCHEMBL932706 0.71 BACE1 (0.66) BACE1CTSDBACE2KCNH2
SCHEMBL932350 0.70 BACE1 (0.50) BACE1CTSDBACE2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed