SCHEMBL9328922

SCHEMBL9328922

Nc1nc(CO/N=C(\[C]=O)c2csc(N)n2)cs1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
GABRA5 P31644 1/20 0.41
GABRB2 P47870 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TP53 P04637 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NOS1 P29475 1/20 0.33
AOC3 Q16853 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136459 0.84 NPC1 (0.34) NPC1RAB9ASMN1; SMN2GABRA5GABRB2
SCHEMBL8136460 0.84 NPC1 (0.34) NPC1RAB9ASMN1; SMN2GABRA5GABRB2
SCHEMBL9367873 0.83 MEN1 (0.41) NPC1RAB9AGABRA5GABRB2HSD17B10
SCHEMBL9143716 0.83 MEN1 (0.41) NPC1RAB9AGABRA5GABRB2HSD17B10
SCHEMBL8316832 0.83 MEN1 (0.51) NPC1RAB9ASMN1; SMN2GABRA5GABRB2
SCHEMBL9329551 0.83 MEN1 (0.41) NPC1RAB9AGABRA5GABRB2HSD17B10
SCHEMBL9331537 0.83 MEN1 (0.41) NPC1RAB9AGABRA5GABRB2HSD17B10
SCHEMBL8316834 0.83 MEN1 (0.51) NPC1RAB9ASMN1; SMN2GABRA5GABRB2
SCHEMBL9143711 0.83 MEN1 (0.41) NPC1RAB9AGABRA5GABRB2HSD17B10
SCHEMBL9332012 0.83 MEN1 (0.51) NPC1RAB9ASMN1; SMN2GABRA5GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0225634-B1 Antibacterial compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1994-04-06 EP disclosed
US-4839351-A Antibacterial compounds, and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-06-13 US disclosed
EP-0229369-A2 Cephalosporins, process for their preparation and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1987-07-22 EP disclosed
EP-0225634-A2 Antibacterial compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-06-16 EP disclosed