SCHEMBL9330875

SCHEMBL9330875

Nc1ccc2nc3ccccc3c(C(=O)O)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.50
PDE10A Q9Y233 3/20 0.50
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.50
GLA P06280 3/20 0.50
HPGD P15428 3/20 0.50
KMT2A Q03164 3/20 0.50
MEN1 O00255 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP1A2 P05177 1/20 0.50
DHODH Q02127 5/20 0.47
LMNA P02545 2/20 0.47
TSHR P16473 2/20 0.46
CASP1 P29466 2/20 0.46
CASP7 P55210 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CHRM2 P08172 1/20 0.46
ADRA2A P08913 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
CHRM1 P11229 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29377848 0.84 PDE10A (0.66) HSD17B10PDE10AKDM4EALDH1A1GLA
SCHEMBL641899 0.84 PDE10A (0.66) HSD17B10PDE10AKDM4EALDH1A1GLA
SCHEMBL17154426 0.82 MDM4 (0.50) HSD17B10PDE10AKDM4EALDH1A1GLA
Water SCHEMBL2991911 0.82 PDE10A (0.63) HSD17B10PDE10AKDM4EALDH1A1GLA
Hydrochloric Acid SCHEMBL1603404 0.82 PDE10A (0.63) HSD17B10PDE10AKDM4EALDH1A1GLA
Iodide SCHEMBL8029606 0.82 PDE10A (0.63) HSD17B10PDE10AKDM4EALDH1A1GLA
Iodide SCHEMBL8029601 0.82 PDE10A (0.63) HSD17B10PDE10AKDM4EALDH1A1GLA
Hydrochloric Acid SCHEMBL9597551 0.82 PDE10A (0.63) HSD17B10PDE10AKDM4EALDH1A1GLA
SCHEMBL3899416 0.81 DHODH (0.55) HSD17B10PDE10AKDM4EALDH1A1GLA
SCHEMBL7698336 0.80 DHODH (0.59) HSD17B10KDM4EALDH1A1GLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0369344-B1 N-arylation of isatins ABBOTT LAB (US) 1994-04-06 EP disclosed
EP-0369344-A1 N-arylation of isatins ABBOTT LABORATORIES (US) 1990-05-23 EP disclosed