SCHEMBL9335752

SCHEMBL9335752

Cc1nc2cnccc2n1-c1cccc(C(=O)O)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.61
THRB P10828 1/20 0.59
HTT P42858 2/20 0.53
TDP1 Q9NUW8 3/20 0.52
KDM4E B2RXH2 2/20 0.52
ALDH1A1 P00352 2/20 0.52
ALOX15 P16050 2/20 0.52
POLB P06746 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
MEN1 O00255 1/20 0.52
USP2 O75604 1/20 0.52
MYC P01106 1/20 0.52
HSPA1A P0DMV8 1/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
NR4A1 P22736 1/20 0.52
PTPN7 P35236 1/20 0.52
RECQL P46063 1/20 0.52
BLM P54132 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7762886 0.85 HSD17B10 (0.72) HSD17B10THRBHTTTDP1KDM4E
SCHEMBL9333280 0.85 ALOX15 (0.62) THRBKDM4EALDH1A1ALOX15MEN1
SCHEMBL7505146 0.84 HSD17B10 (0.59) HSD17B10THRBHTTTDP1KDM4E
SCHEMBL7876035 0.81 ALOX15 (0.48) HSD17B10THRBALOX15MEN1KMT2A
SCHEMBL4446308 0.81 MRGPRX4 (0.58) HSD17B10THRBSMN1; SMN2PKM
SCHEMBL9524668 0.81 HSD17B10 (0.55) HSD17B10HTTMEN1KMT2ASMN1; SMN2
SCHEMBL540767 0.81 MAPK1 (0.67) HSD17B10HTTKDM4EALDH1A1SMN1; SMN2
SCHEMBL13243754 0.78 HSD17B10 (0.65) HSD17B10THRBHTTTDP1KDM4E
SCHEMBL1356522 0.77 HSD17B10 (0.64) HSD17B10THRBHTTTDP1KDM4E
SCHEMBL12135360 0.77 HSD17B10 (0.64) HSD17B10THRBHTTTDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5358953-A For treatment of allergic rhinitis PFIZER INC. (US) 1994-10-25 US disclosed
EP-0572425-B1 IMIDAZOPYRIDINE PAF/H 1 ANTAGONISTS PFIZER LTD (GB) 1994-08-03 EP disclosed
EP-0572425-A1 IMIDAZOPYRIDINE PAF/H 1? ANTAGONISTS. PFIZER LTD (GB) 1993-12-08 EP disclosed
WO-1992014734-A1 IMIDAZOPYRIDINE PAF/H1 ANTAGONISTS PFIZER LIMITED (GB) 1992-09-03 WO disclosed