SCHEMBL933832

SCHEMBL933832

CC(Cc1ccc(I)cc1)C(N)=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.49
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
APEX1 P27695 1/20 0.46
PMP22 Q01453 1/20 0.46
DPP4 P27487 2/20 0.40
ALOX5 P09917 2/20 0.40
DPP7 Q9UHL4 1/20 0.38
TAAR1 Q96RJ0 2/20 0.38
SLC6A2 P23975 1/20 0.38
LMNA P02545 1/20 0.38
ALB P02768 1/20 0.38
ESR1 P03372 1/20 0.38
RARB P10826 1/20 0.38
CYP2C9 P11712 1/20 0.38
ADRB3 P13945 1/20 0.38
NFKB1 P19838 1/20 0.38
PTGS1 P23219 1/20 0.38
HTR2A P28223 1/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14019341 0.82 CYP1A2 (0.48) CYP1A2CYP2D6APEX1PMP22DPP4
SCHEMBL14032489 0.82 TAAR1 (0.59) EPHX1TAAR1SLC6A2ESR1
SCHEMBL22937469 0.82 EPHX1 (0.50) EPHX1PMP22ALOX5TAAR1SLC6A2
SCHEMBL23643109 0.82 EPHX1 (0.50) EPHX1CYP2D6ALOX5TAAR1SLC6A2
SCHEMBL934530 0.82 TAAR1 (0.59) EPHX1TAAR1SLC6A2ESR1
SCHEMBL23643108 0.82 EPHX1 (0.50) EPHX1ALOX5TAAR1SLC6A2
SCHEMBL12639935 0.82 TBXAS1 (0.51) CYP1A2CYP2D6APEX1PMP22ALOX5
SCHEMBL22593510 0.82 EPHX1 (0.50) EPHX1DPP4ALOX5TAAR1
SCHEMBL457465 0.82 TBXAS1 (0.51) CYP1A2CYP2D6APEX1PMP22ALOX5
SCHEMBL12118748 0.82 EPHX1 (0.50) EPHX1DPP4ALOX5TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011037833-A2 NOVEL N-BENZYLAMIDE SUBSTITUTED DERIVATIVES OF 2-(ACYLAMIDO)ACETIC ACID AND 2-(ACYLAMIDO)PROPIONIC ACIDS: POTENT NEUROLOGICAL AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2011-03-31 WO disclosed
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed