SCHEMBL9341876

SCHEMBL9341876

CCc1c(C(=O)O)c(=O)c2cc(F)c(Cl)cc2n1CC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 10/20 0.50
PIM2 Q9P1W9 5/20 0.50
GSK3A P49840 2/20 0.50
PIM3 Q86V86 1/20 0.50
DAPK3 O43293 1/20 0.37
MET P08581 1/20 0.37
KDR P35968 1/20 0.37
CSNK1D P48730 1/20 0.37
RPS6KA3 P51812 1/20 0.37
CSNK2A1 P68400 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PAK1 Q13153 1/20 0.37
STK3 Q13188 1/20 0.37
DYRK1A Q13627 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
DRD3 P35462 1/20 0.35
GRIA1 P42261 1/20 0.35
GRIA2 P42262 1/20 0.35
GRIA3 P42263 1/20 0.35
GRIA4 P48058 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20527932 0.83 PIM1 (0.48) PIM1PIM2GSK3APIM3RPS6KA3
SCHEMBL9748506 0.83 PIM1 (0.38) PIM1PIM2GSK3APIM3RPS6KA3
SCHEMBL9715578 0.81 KDM4E (0.39) PIM1PIM2GSK3APIM3RPS6KA3
SCHEMBL10623503 0.81 KDM4E (0.35) PIM1PIM2GSK3APIM3DRD3
SCHEMBL10620783 0.81 HPGD (0.35) PIM1PIM2GSK3APIM3DRD3
SCHEMBL11096126 0.81 DRD3 (0.39) PIM1GSK3APIM3RPS6KA3DYRK1A
SCHEMBL10427396 0.80 CCR3 (0.37) PIM1PIM2GSK3APIM3KDM4E
SCHEMBL9151598 0.80 GSK3B (0.44) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL9748573 0.79 PIM1 (0.36) PIM1PIM2GSK3APIM3DRD3
SCHEMBL10553019 0.78 PIM1 (0.35) PIM1PIM2GSK3APIM3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0351889-B1 Process for the preparation of a quinoline carboxylic acid CHINOIN GYOGYSZER ES VEGYESZET (HU) 1994-06-29 EP disclosed
US-5294712-A Process for the preparation of quinoline carboxylic acids CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1994-03-15 US disclosed
US-5284950-A Process for the preparation of quinoline carboxyolic acids CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1994-02-08 US disclosed
EP-0249620-B1 PROCESS FOR THE PREPARATION OF QUINOLINE CARBOXYLIC ACIDS CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1992-11-19 EP disclosed
US-4981966-A Process for the preparation of quinoline carboxylic acids CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1991-01-01 US disclosed
EP-0250535-B1 NORFLOXACIN INTERMEDIATE CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1990-05-30 EP disclosed
EP-0351889-A1 Process for the preparation of a quinoline carboxylic acid CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1990-01-24 EP disclosed
US-4803274-A Norfloxacin intermediate CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1989-02-07 US disclosed
EP-0250535-A1 NORFLOXACIN INTERMEDIATE. CHINOIN GYOGYSZER ES VEGYESZET (HU) 1988-01-07 EP disclosed
EP-0249620-A1 PROCESS FOR THE PREPARATION OF QUINOLINE CARBOXYLIC ACIDS. CHINOIN GYOGYSZER ES VEGYESZET (HU) 1987-12-23 EP disclosed
WO-1987003587-A1 PROCESS FOR THE PREPARATION OF QUINOLINE CARBOXYLIC ACIDS Chinoin Gyógyszer és Vegyészeti Termékek Gyára Rt. (HU) 1987-06-18 WO disclosed
WO-1987003595-A1 NORFLOXACIN INTERMEDIATE Chinoin Gyógyszer és Vegyészeti Termékek Gyára Rt. (HU) 1987-06-18 WO disclosed