SCHEMBL934416

SCHEMBL934416

COC(=O)CCN(C(=O)OC(C)(C)C)[C@@H](CC(=O)OC)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CA12 O43570 2/20 0.38
CA2 P00918 2/20 0.38
CA1 P00915 1/20 0.38
SLC1A1 P43005 1/20 0.34
TSHR P16473 3/20 0.33
GAA P10253 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
TDP1 Q9NUW8 1/20 0.30
SELP P16109 1/20 0.30
REN P00797 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5837182 1.00 CA14 (0.38) CA14MEN1KMT2ACA12CA2
SCHEMBL23854196 1.00 CA14 (0.38) CA14MEN1KMT2ACA12CA2
SCHEMBL4547485 0.89 CA14 (0.38) CA14MEN1KMT2ACA12CA2
SCHEMBL17881260 0.82 MEN1 (0.40) CA14MEN1KMT2ACA12CA2
SCHEMBL21385385 0.82 MEN1 (0.40) CA14MEN1KMT2ACA12CA2
SCHEMBL13345432 0.81 MAPT (0.33) CA14MEN1KMT2ACA12CA2
SCHEMBL3899118 0.80 REN (0.40) CA14MEN1KMT2ACA12CA2
SCHEMBL13598307 0.80 REN (0.40) CA14MEN1KMT2ACA12CA2
SCHEMBL18248185 0.80 REN (0.40) CA14MEN1KMT2ACA12CA2
SCHEMBL20593366 0.80 CA14 (0.38) CA14MEN1KMT2ACA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250136620-A1 BTK DEGRADER NEWAVE PHARMACEUTICAL INC. 2025-05-01 US disclosed
EP-4263552-A1 BTK DEGRADER Guangzhou Lupeng Pharmaceutical Company Ltd. (CN) 2023-10-25 EP disclosed
WO-2023137225-A1 BTK DEGRADER NEWAVE PHARMACEUTICAL INC. (US) 2023-07-20 WO disclosed
WO-2022133184-A1 BTK DEGRADER NEWAVE PHARMACEUTICAL INC. (US) 2022-06-23 WO disclosed
WO-2022133184-A1 BTK DEGRADER NEWAVE PHARMACEUTICAL INC. (US) 2022-06-23 WO disclosed
CN-102471314-B Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction ROTTAPHARM SPA 2015-05-13 CN disclosed
EP-2454252-B1 Spiro amino compounds suitable for the treatment of (inter alia) sleep disorders and drug addiction Rottapharm Biotech Srl (IT) 2015-03-04 EP disclosed
EP-2454252-B1 Spiro amino compounds suitable for the treatment of (inter alia) sleep disorders and drug addiction Rottapharm Biotech Srl (IT) 2015-03-04 EP disclosed
US-8859608-B2 Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction ROTTAPHARM BIOTECH S.R.L. (IT) 2014-10-14 US disclosed
US-8859608-B2 Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction ROTTAPHARM BIOTECH S.R.L. (IT) 2014-10-14 US disclosed
EP-2454252-A1 SPIRO AMINO COMPOUNDS SUITABLE FOR THE TREATMENT OF INTER ALIA SLEEP DISORDERS AND DRUG ADDICTION Rottapharm S.p.A. (IT) 2012-05-23 EP disclosed
CN-102471314-A Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction ROTTAPHARM SPA 2012-05-23 CN disclosed
US-20120115882-A1 SPIRO AMINO COMPOUNDS SUITABLE FOR THE TREATMENT OF INTER ALIA SLEEP DISORDERS AND DRUG ADDICTION ROTTAPHARM BIOTECH S.R.L. (IT) 2012-05-10 US disclosed
US-20120115882-A1 SPIRO AMINO COMPOUNDS SUITABLE FOR THE TREATMENT OF INTER ALIA SLEEP DISORDERS AND DRUG ADDICTION ROTTAPHARM BIOTECH S.R.L. (IT) 2012-05-10 US disclosed
WO-2011006960-A1 SPIRO AMINO COMPOUNDS SUITABLE FOR THE TREATMENT OF INTER ALIA SLEEP DISORDERS AND DRUG ADDICTION ROTTAPHARM S.P.A. (IT) 2011-01-20 WO disclosed
WO-2011006960-A1 SPIRO AMINO COMPOUNDS SUITABLE FOR THE TREATMENT OF INTER ALIA SLEEP DISORDERS AND DRUG ADDICTION ROTTAPHARM S.P.A. (IT) 2011-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120115882-A1 SPIRO AMINO COMPOUNDS SUITABLE FOR THE TREATMENT OF INTER ALIA SLEEP DISORDERS AND DRUG ADDICTION SLC1A1, SLC6A3, SLC1A2 CA14 3870/4885MEN1 2457/4885KMT2A 108/4885
US-20250136620-A1 BTK DEGRADER BTK, CBL, LYN CA14 4242/4885MEN1 2462/4885KMT2A 549/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.