Cycloheximide

Cycloheximide

SCHEMBL9344504

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nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

FAURPL10RPL10ARPL11RPL12RPL13RPL13ARPL14RPL15RPL17RPL18RPL18ARPL19RPL21RPL22RPL23RPL23ARPL24RPL26RPL27RPL27ARPL28RPL29RPL3RPL30RPL31RPL32RPL34RPL35RPL35ARPL36RPL36ARPL37RPL37ARPL38RPL39RPL4RPL41RPL5RPL6RPL7RPL7ARPL8RPL9RPL9P7RPL9P8RPL9P9RPLP0RPLP1RPS10RPS11RPS12RPS13RPS14RPS15RPS15ARPS16RPS17RPS18RPS19RPS2RPS20RPS21RPS23RPS24RPS25RPS26RPS27RPS27ARPS28RPS29RPS3RPS3ARPS4XRPS4Y1RPS5RPS6RPS7RPS8RPS9RPSA

The experimentally established mechanism targets of Cycloheximide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 10/20 1.00
SMN1; SMN2 Q16637 4/20 1.00
NR2F2 P24468 3/20 1.00
ALDH1A1 P00352 3/20 1.00
LMNA P02545 2/20 1.00
NPC1 O15118 2/20 1.00
RAB9A P51151 2/20 1.00
HIF1A Q16665 2/20 1.00
FKBP4 Q02790 2/20 1.00
CYP1A2 P05177 1/20 1.00
CYP2C19 P33261 1/20 1.00
MAPK1 P28482 1/20 1.00
TP53 P04637 1/20 1.00
CYP3A4 P08684 1/20 1.00
SLC2A1 P11166 1/20 1.00
EIF4A1 P60842 1/20 1.00
EPAS1 Q99814 1/20 1.00
FKBP14 Q9NWM8 1/20 1.00
HTT P42858 1/20 1.00
FKBP5 Q13451 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cycloheximide SCHEMBL30020292 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Cycloheximide SCHEMBL1714687 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Cycloheximide SCHEMBL3764340 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Naramycin B SCHEMBL29356383 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Cycloheximide SCHEMBL1753509 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Cycloheximide SCHEMBL17223570 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Cycloheximide SCHEMBL24914327 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Cycloheximide SCHEMBL674135 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Cycloheximide SCHEMBL26617 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA
Cycloheximide SCHEMBL3764335 1.00 FKBP1A (1.00) FKBP1ASMN1; SMN2NR2F2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108624621-B The preparation method of the somatic cell clone animal of non-human primates 中国科学院上海生命科学研究院 2019-04-12 CN claimed
CN-116459332-B Mechanism for promoting autophagy of cells by using ubiquitinated stable Rab7a of OTUD3 protein and application of mechanism 中国人民解放军军事科学院军事医学研究院 2023-10-13 CN disclosed
CN-116459332-A Mechanism for promoting autophagy of cells by using ubiquitinated stable Rab7a of OTUD3 protein and application of mechanism 中国人民解放军军事科学院军事医学研究院 2023-07-21 CN disclosed
CN-108624621-B The preparation method of the somatic cell clone animal of non-human primates 中国科学院上海生命科学研究院 2019-04-12 CN disclosed
CN-108624621-A The preparation method of the somatic cell clone animal of non-human primates 中国科学院上海生命科学研究院 2018-10-09 CN disclosed
US-9658229-B2 Modulators of itch ubiquitinase activity RYBOQUIN COMPANY LIMITED (GB) 2017-05-23 US disclosed
CN-103911368-B Based on immuno-precipitation from Oryza sativa L., extract polysomal method 复旦大学 2016-08-17 CN disclosed
US-20160084838-A1 Modulators of Itch Ubiquitinase Activity MEDICAL RESEARCH COUNCIL (GB) 2016-03-24 US disclosed
WO-2014172616-A2 METHODS, COMPOSITIONS AND KITS FOR PROMOTING MOTOR NEURON SURVIVAL AND TREATING AND DIAGNOSING NEURODEGENERATIVE DISORDERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2014-10-23 WO disclosed
CN-103911368-A Method for extracting polysome from rice on basis of immune-precipitation UNIV FUDAN 2014-07-09 CN disclosed
US-5296358-A Oxidative deamination MINISTERO DELL'UNIVERSITA' E DELLA RICERCA SCIENTIFICA E TECNOLOGICA (IT) 1994-03-22 US disclosed