SCHEMBL934552

SCHEMBL934552

NC(=O)CCCc1cccc(OC(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.51
CHRM1 P11229 1/20 0.51
CHRM3 P20309 1/20 0.51
CNR1 P21554 1/20 0.50
DAO P14920 1/20 0.50
EPHX1 P07099 1/20 0.49
TRPM8 Q7Z2W7 1/20 0.48
FFAR1 O14842 1/20 0.48
PPARG P37231 2/20 0.48
PPARA Q07869 2/20 0.48
MAPK14 Q16539 1/20 0.47
PLA2G10 O15496 1/20 0.47
PLA2G2A P14555 1/20 0.47
PLA2G5 P39877 1/20 0.47
CETP P11597 1/20 0.46
FFAR4 Q5NUL3 1/20 0.46
AMPD2 Q01433 1/20 0.46
ROCK2 O75116 1/20 0.44
ROCK1 Q13464 1/20 0.44
GRIN2B Q13224 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL934428 0.94 PPARG (0.52) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL5724443 0.93 CHRM2 (0.52) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL30487710 0.93 CHRM2 (0.52) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL15818310 0.88 FFAR1 (0.57) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL17261637 0.84 FFAR1 (0.56) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL27997591 0.83 CHRM2 (0.55) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL6685564 0.83 EPHX1 (0.52) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL4981663 0.83 TRPM8 (0.49) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL15818398 0.82 PPARA (0.55) CHRM2CHRM1CHRM3CNR1DAO
SCHEMBL1271844 0.82 FFAR1 (0.67) CHRM2CHRM1CHRM3CNR1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1780821-A Heterocyclic kinase inhibitors. ABBOTT LAB (US) 2006-05-31 CN claimed
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed
CN-1780821-A Heterocyclic kinase inhibitors. ABBOTT LAB (US) 2006-05-31 CN disclosed