SCHEMBL934428

SCHEMBL934428

NC(=O)CCCCCc1cccc(OC(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.52
PPARA Q07869 4/20 0.52
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
EPHX1 P07099 1/20 0.50
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
CHRM3 P20309 1/20 0.49
FAAH O00519 3/20 0.49
CES1 P23141 3/20 0.49
CNR1 P21554 1/20 0.48
DAO P14920 1/20 0.48
TRPM8 Q7Z2W7 1/20 0.46
FFAR1 O14842 1/20 0.46
MAPK14 Q16539 1/20 0.45
PLA2G10 O15496 1/20 0.45
PLA2G2A P14555 1/20 0.45
PLA2G5 P39877 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL934552 0.94 CHRM2 (0.51) PPARGPPARAEPHX1CHRM2CHRM1
SCHEMBL30487710 0.90 CHRM2 (0.52) EPHX1CHRM2CHRM1CHRM3CNR1
SCHEMBL5724443 0.90 CHRM2 (0.52) EPHX1CHRM2CHRM1CHRM3CNR1
SCHEMBL17261637 0.87 FFAR1 (0.56) PPARGPPARAHDAC1HDAC6CHRM2
SCHEMBL17261656 0.84 HDAC1 (0.54) PPARGPPARAHDAC1HDAC6CHRM2
SCHEMBL15818310 0.83 FFAR1 (0.57) PPARGPPARAHDAC1HDAC6CHRM2
SCHEMBL934358 0.82 FAAH (0.51) PPARAHDAC1HDAC6EPHX1FAAH
SCHEMBL6232367 0.82 CHRM2 (0.50) PPARGPPARACHRM2CHRM1CHRM3
SCHEMBL12040546 0.82 PPARG (0.52) PPARGPPARACHRM2CHRM1CHRM3
SCHEMBL934608 0.81 HDAC1 (0.72) HDAC1HDAC6CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed