SCHEMBL9347398

SCHEMBL9347398

CCc1cc2[nH]c(=O)c(-c3ccccc3)cc2c(CC)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48
ATM Q13315 1/20 0.48
KDM4E B2RXH2 3/20 0.44
PKM P14618 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MAT2A P31153 1/20 0.39
TP53 P04637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CHEK1 O14757 1/20 0.39
TNKS2 Q9H2K2 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
HPGD P15428 2/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
LYN P07948 1/20 0.37
SRC P12931 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9346570 0.86 HPGD (0.45) KMT2AKDM4EHPGDALDH1A1CDK5
SCHEMBL9346657 0.82 LMNA (0.45) NPC1RAB9AATMKDM4EPKM
SCHEMBL9347480 0.81 KDM4E (0.42) KDM4EPKMTDP1SMN1; SMN2TNKS2
SCHEMBL9346549 0.79 BRD4 (0.40) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL9347518 0.78 KDM4E (0.39) MEN1KMT2AKDM4EPKMTDP1
SCHEMBL9347456 0.75 PLK4 (0.46) KDM4ETDP1SMN1; SMN2CHEK1HPGD
SCHEMBL9347463 0.74 PDE3B (0.41) KMT2AKDM4EHPGDMAPK1ALDH1A1
SCHEMBL9346572 0.74 GAA (0.43) KDM4EHPGD
SCHEMBL3179823 0.74 PDE3B (0.58) KDM4ESMN1; SMN2MAT2ATP53HPGD
SCHEMBL3177677 0.73 NPC1 (0.51) MEN1NPC1RAB9AKMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294620-A Hypotensive agents or compounds for cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-03-15 US disclosed
US-5217976-A Hypotensive agents, congestive heart failure IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-06-08 US disclosed