SCHEMBL9350672

SCHEMBL9350672

CCCn1cnc2c1c(=O)n(CC1CCC1)c(=O)n2CC1CCC1

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 12/20 0.60
PDE4B Q07343 12/20 0.60
PDE4C Q08493 12/20 0.60
PDE4D Q08499 12/20 0.60
ADORA2A P29274 8/20 0.60
ADORA2B P29275 7/20 0.60
PDE5A O76074 1/20 0.53
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9350638 0.95 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9350777 0.83 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9350631 0.83 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9350653 0.82 SMN1; SMN2 (0.54) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9350644 0.82 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL316171 0.81 PDE4A (0.82) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9350645 0.81 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9350699 0.80 SMN1; SMN2 (0.54) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9350756 0.80 PDE4A (0.59) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9350791 0.79 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0369744-B1 Xanthine derivatives, process for their preparation and pharmaceutical compositions SMITHKLINE BEECHAM PHARMA GMBH (DE) 1994-09-21 EP claimed
US-5321029-A Vascular and skin disorders; bronchodilator BEECHAM-WUELFING GMBH & CO.K.G. (DE) 1994-06-14 US claimed
EP-0369744-A2 Xanthine derivatives, process for their preparation and pharmaceutical compositions SMITHKLINE BEECHAM PHARMA GmbH (DE) 1990-05-23 EP claimed
EP-0369744-B1 Xanthine derivatives, process for their preparation and pharmaceutical compositions SMITHKLINE BEECHAM PHARMA GMBH (DE) 1994-09-21 EP disclosed
US-5321029-A Vascular and skin disorders; bronchodilator BEECHAM-WUELFING GMBH & CO.K.G. (DE) 1994-06-14 US disclosed
EP-0369744-A2 Xanthine derivatives, process for their preparation and pharmaceutical compositions SMITHKLINE BEECHAM PHARMA GmbH (DE) 1990-05-23 EP disclosed