SCHEMBL9356145

SCHEMBL9356145

CC(=O)Oc1ccc(C(=O)CN2CCN(C)CC2)cc1OC(C)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.51
KDM4E B2RXH2 4/20 0.51
GAA P10253 2/20 0.51
TSHR P16473 2/20 0.51
RAB9A P51151 1/20 0.51
MAPT P10636 4/20 0.49
CYP2D6 P10635 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
POLB P06746 1/20 0.49
CNR2 P34972 1/20 0.46
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
HTT P42858 1/20 0.45
ALOX15 P16050 1/20 0.44
TOP1 P11387 1/20 0.44
HPGD P15428 2/20 0.43
RECQL P46063 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9012958 0.79 KMT2A (0.56) ALDH1A1KDM4EGAATSHRRAB9A
SCHEMBL13981872 0.78 ACHE (0.42) ALDH1A1KDM4EGAATSHRRAB9A
SCHEMBL9356659 0.76 ALPG (0.70) ALDH1A1KDM4EGAAMAPTPOLB
SCHEMBL20033130 0.74 PDE4B (0.44) ALDH1A1KDM4EMAPTCYP2D6CYP1A2
SCHEMBL26921558 0.74 ALDH1A1 (0.60) ALDH1A1KDM4EGAATSHRRAB9A
SCHEMBL11837908 0.74 ALDH1A1 (0.50) ALDH1A1KDM4EGAAMAPTCYP2D6
SCHEMBL11111092 0.73 TSHR (0.64) ALDH1A1KDM4EGAATSHRRAB9A
SCHEMBL2616297 0.73 KMT2A (0.76) ALDH1A1KDM4ETSHRCYP1A2CYP2C19
SCHEMBL9198139 0.73 ALDH1A1 (0.64) ALDH1A1KDM4EGAATSHRRAB9A
SCHEMBL9651777 0.73 TSHR (0.64) ALDH1A1KDM4EGAATSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0416410-B1 Piperaziniocephalosporins SHIONOGI & CO (JP) 1994-11-30 EP disclosed
US-5143910-A PIPERAZINIOCEPHALOSPORINS SHIONOGI & CO., LTD. (JP) 1992-09-01 US disclosed
EP-0416410-A1 Piperaziniocephalosporins SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1991-03-13 EP disclosed