SCHEMBL9357019

SCHEMBL9357019

O=[PH](O)CCCCCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.55
RXFP1 Q9HBX9 1/20 0.55
HDAC1 Q13547 4/20 0.49
HDAC2 Q92769 2/20 0.49
ALOX5 P09917 1/20 0.49
SIGMAR1 Q99720 6/20 0.48
HDAC3 O15379 1/20 0.48
MAPK1 P28482 1/20 0.48
ADRA1A P35348 1/20 0.48
HDAC4 P56524 1/20 0.48
SLC6A3 Q01959 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
FAAH O00519 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25331935 1.00 MAPT (0.55) MAPTRXFP1HDAC1HDAC2ALOX5
SCHEMBL25332105 1.00 MAPT (0.55) MAPTRXFP1HDAC1HDAC2ALOX5
SCHEMBL7931539 1.00 MAPT (0.55) MAPTRXFP1HDAC1HDAC2ALOX5
SCHEMBL28910960 0.98 MAPT (0.53) MAPTRXFP1HDAC1HDAC2ALOX5
SCHEMBL2357339 0.98 MAPT (0.52) MAPTRXFP1HDAC1HDAC2ALOX5
SCHEMBL28539291 0.96 MAPT (0.50) MAPTRXFP1HDAC1HDAC2ALOX5
SCHEMBL3822270 0.92 HDAC3 (0.52) MAPTRXFP1HDAC1HDAC2SIGMAR1
SCHEMBL28529981 0.90 HDAC3 (0.50) MAPTRXFP1HDAC1HDAC2SIGMAR1
SCHEMBL7931875 0.90 HDAC3 (0.50) MAPTRXFP1HDAC1HDAC2SIGMAR1
SCHEMBL942065 0.83 KEAP1 (0.48) MAPTRXFP1HDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478624-B Telomer of diethyl aluminum phosphinate and preparation method thereof 兰州瑞朴科技有限公司 2024-07-02 CN claimed
WO-2023138015-A1 ALUMINUM DIETHYLPHOSPHINATE FLAME RETARDANT AND PREPARATION METHOD THEREFOR 兰州瑞朴科技有限公司 2023-07-27 WO claimed
CN-114478624-A Telomer of aluminum diethylphosphinate and preparation method thereof 兰州瑞朴科技有限公司 2022-05-13 CN claimed
CN-115109310-B Flame retardant and corresponding flame-retardant plastic product 兰州瑞朴科技有限公司 2024-07-02 CN disclosed
CN-114478624-B Telomer of diethyl aluminum phosphinate and preparation method thereof 兰州瑞朴科技有限公司 2024-07-02 CN disclosed
WO-2023138015-A1 ALUMINUM DIETHYLPHOSPHINATE FLAME RETARDANT AND PREPARATION METHOD THEREFOR 兰州瑞朴科技有限公司 2023-07-27 WO disclosed
CN-112778511-B Catalyst composition for polyester production process 科莱恩塑料和涂料有限公司 2023-03-28 CN disclosed
CN-115109310-A Flame retardant and corresponding flame-retardant plastic product 兰州瑞朴科技有限公司 2022-09-27 CN disclosed
CN-114478624-A Telomer of aluminum diethylphosphinate and preparation method thereof 兰州瑞朴科技有限公司 2022-05-13 CN disclosed
CN-112778511-A Catalyst composition for polyester production process 科莱恩塑料和涂料有限公司 2021-05-11 CN disclosed
CN-107075097-B Catalyst composition for polyester production process 科莱恩塑料和涂料有限公司 2021-02-05 CN disclosed
EP-0350138-B1 Processes for preparing phosphonyl hydroxyacyl prolines SQUIBB & SONS INC (US) 1994-10-19 EP disclosed
EP-0350138-A2 Processes for preparing phosphonyl hydroxyacyl prolines E.R. SQUIBB & SONS, INC. (US) 1990-01-10 EP disclosed
EP-0138403-B1 PROCESS FOR PREPARING PHOSPHINIC ACID INTERMEDIATES E.R. Squibb & Sons, Inc. (US) 1989-03-15 EP disclosed
US-4745196-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1988-05-17 US disclosed
EP-0229520-A1 Orally active phosphonyl hydroxyacyl prolines and processes for preparing phosphonyl hydroxyacyl prolines E.R. Squibb & Sons, Inc. (US) 1987-07-22 EP disclosed
EP-0138403-A2 Process for preparing phosphinic acid intermediates E.R. Squibb & Sons, Inc. (US) 1985-04-24 EP disclosed