SCHEMBL936381

SCHEMBL936381

CC(C)NCC(O)c1ccc(-c2cc(-c3cccc(C(=O)NC(C)C#N)c3)no2)cc1

nearest known ligand 0.77

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 11/20 0.77
PRKD3 O94806 1/20 0.61
PRKD2 Q9BZL6 1/20 0.61
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PPARG P37231 2/20 0.38
PPARA Q07869 2/20 0.38
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
MLLT1 Q03111 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL936379 1.00 PRKD1 (0.77) PRKD1PRKD3PRKD2ALDH1A1NPC1
SCHEMBL935843 0.87 PRKD1 (1.00) PRKD1PRKD3PRKD2ALDH1A1NPC1
SCHEMBL935844 0.87 PRKD1 (1.00) PRKD1PRKD3PRKD2ALDH1A1NPC1
SCHEMBL937700 0.85 PRKD1 (0.54) PRKD1PRKD3PRKD2NPC1RAB9A
SCHEMBL935842 0.84 PRKD1 (0.69) PRKD1PRKD3PRKD2ALDH1A1NPC1
SCHEMBL938420 0.84 PRKD1 (0.81) PRKD1PRKD3PRKD2ALDH1A1NPC1
SCHEMBL938421 0.84 PRKD1 (0.81) PRKD1PRKD3PRKD2ALDH1A1NPC1
SCHEMBL6922430 0.83 PRKD1 (0.52) PRKD1PRKD3PRKD2ALDH1A1NPC1
SCHEMBL935481 0.82 PRKD1 (0.72) PRKD1PRKD3PRKD2ALDH1A1NPC1
SCHEMBL935480 0.82 PRKD1 (0.72) PRKD1PRKD3PRKD2ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009484-A1 ARYLPYRAZOLES AND ARYLISOXAZOLES AND THEIR USE AS PKD MODULATORS NOVARTIS AG (CH) 2011-01-27 WO disclosed