SCHEMBL9364141

SCHEMBL9364141

COc1ccc(/C=C/C(=O)N2CCOCC2)cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.81
KDM4E B2RXH2 7/20 0.78
ALDH1A1 P00352 4/20 0.78
KMT2A Q03164 3/20 0.78
L3MBTL1 Q9Y468 1/20 0.74
HPGD P15428 3/20 0.74
SMN1; SMN2 Q16637 2/20 0.74
APP P05067 2/20 0.74
MEN1 O00255 2/20 0.74
TDP1 Q9NUW8 2/20 0.70
NPC1 O15118 1/20 0.62
RAB9A P51151 1/20 0.62
ITGB2 P05107 1/20 0.62
ICAM1 P05362 1/20 0.62
ITGAL P20701 1/20 0.62
MAOB P27338 2/20 0.61
BCHE P06276 1/20 0.61
MAOA P21397 1/20 0.61
ACHE P22303 1/20 0.61
PTGS2 P35354 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9363901 1.00 TRPV1 (0.81) TRPV1KDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL2122038 0.90 TRPV1 (1.00) TRPV1KDM4EALDH1A1KMT2AHPGD
SCHEMBL2122045 0.90 TRPV1 (1.00) TRPV1KDM4EALDH1A1KMT2AHPGD
SCHEMBL8077987 0.87 TRPV1 (0.66) TRPV1KDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL8077994 0.87 TRPV1 (0.66) TRPV1KDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL15110739 0.87 TRPV1 (0.69) TRPV1KDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL15110741 0.87 TRPV1 (0.69) TRPV1KDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL3121297 0.86 KDM4E (0.97) TRPV1KDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL3121290 0.86 KDM4E (0.97) TRPV1KDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL11469833 0.85 KDM4E (0.80) TRPV1KDM4EALDH1A1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0219756-B1 Acrylic amides SHELL INT RESEARCH (NL) 1994-01-05 EP claimed
EP-0219756-A1 Acrylic amides SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1987-04-29 EP claimed
EP-0219756-B1 Acrylic amides SHELL INT RESEARCH (NL) 1994-01-05 EP disclosed
US-4910200-A Agricultural fungicide CELAMERCK GMBH & CO. KG (DE) 1990-03-20 US disclosed
EP-0219756-A1 Acrylic amides SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1987-04-29 EP disclosed