SCHEMBL8077987

SCHEMBL8077987

CCCCCOc1cc(/C=C/C(=O)N2CCOCC2)ccc1OC

nearest known ligand 0.90

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.66
KDM4E B2RXH2 5/20 0.64
KMT2A Q03164 3/20 0.64
APP P05067 3/20 0.64
HPGD P15428 2/20 0.64
MEN1 O00255 2/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
TDP1 Q9NUW8 1/20 0.60
ALDH1A1 P00352 2/20 0.60
L3MBTL1 Q9Y468 1/20 0.57
THRB P10828 1/20 0.54
CNR2 P34972 2/20 0.52
ITGB2 P05107 1/20 0.52
ICAM1 P05362 1/20 0.52
ITGAL P20701 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8077994 1.00 TRPV1 (0.66) TRPV1KDM4EKMT2AAPPHPGD
SCHEMBL9363901 0.87 TRPV1 (0.81) TRPV1KDM4EKMT2AAPPHPGD
SCHEMBL9364141 0.87 TRPV1 (0.81) TRPV1KDM4EKMT2AAPPHPGD
SCHEMBL4409428 0.82 KDM4E (0.80) KDM4EHPGDSMN1; SMN2ALDH1A1CNR2
SCHEMBL4409431 0.82 KDM4E (0.80) KDM4EHPGDSMN1; SMN2ALDH1A1CNR2
SCHEMBL14441230 0.80 RAB9A (0.91) TRPV1KDM4EKMT2AHPGDMEN1
SCHEMBL2122038 0.80 TRPV1 (1.00) TRPV1KDM4EKMT2AAPPHPGD
SCHEMBL2122045 0.80 TRPV1 (1.00) TRPV1KDM4EKMT2AAPPHPGD
SCHEMBL8085980 0.80 KDM4E (0.76) KDM4EKMT2AHPGDSMN1; SMN2ALDH1A1
SCHEMBL8085985 0.80 KDM4E (0.76) KDM4EKMT2AHPGDSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017919-A Compounds and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2000-01-25 US disclosed
EP-0887340-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL USE THEREOF Japan Tobacco Inc. (JP) 1998-12-30 EP disclosed