SCHEMBL9364256

SCHEMBL9364256

CCCCOC(=O)OC1=C(C)N(C2CC2)C(C)=C(OC(=O)OC)C1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ATM Q13315 1/20 0.36
LIPC P11150 1/20 0.36
LIPG Q9Y5X9 1/20 0.36
NOD2 Q9HC29 3/20 0.35
NOD1 Q9Y239 3/20 0.35
ACHE P22303 2/20 0.35
BCHE P06276 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
SLC6A5 Q9Y345 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9367612 0.94 KDM4E (0.41) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9363990 0.91 ALDH1A1 (0.47) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9364676 0.89 KDM4E (0.53) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9363819 0.88 KDM4E (0.42) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9364594 0.88 KDM4E (0.42) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9363848 0.87 KDM4E (0.46) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9364022 0.83 KDM4E (0.41) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9364015 0.82 HSP90AA1 (0.42) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9122411 0.82 GAA (0.51) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL9446688 0.79 KDM4E (0.45) KDM4EALDH1A1POLBGAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0451654-B1 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1994-09-07 EP claimed
EP-0451654-A2 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1991-10-16 EP claimed
EP-0451654-B1 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1994-09-07 EP disclosed
EP-0451654-A2 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1991-10-16 EP disclosed